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A Pore Segment in DEG/ENaC Na+Channels
Journal article   Open access   Peer reviewed

A Pore Segment in DEG/ENaC Na+Channels

Peter M Snyder, Diane R Olson and Daniel B Bucher
The Journal of biological chemistry, Vol.274(40), pp.28484-28490
10/01/1999
DOI: 10.1074/jbc.274.40.28484
PMID: 10497211
url
https://doi.org/10.1074/jbc.274.40.28484View
Published (Version of record) Open Access

Abstract

DEG/ENaC Na(+) channels have diverse functions, including Na(+) absorption, neurotransmission, and sensory transduction. The ability of these channels to discriminate between different ions is critical for their normal function. Several findings suggest that DEG/ENaC channels have a pore structure similar to K(+) channels. To test this hypothesis, we examined the accessibility of native and introduced cysteines in the putative P loop of ENaC. We identified residues that span a barrier that excludes amiloride as well as anionic and large methanethiosulfonate reagents from the pore. This segment contains a structural element ((S/G)CS) involved in selectivity of ENaC. The results are not consistent with predictions from the K(+) channel pore, suggesting that DEG/ENaC Na(+) channels have a novel pore structure.

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