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Characterization of the PNT1 pentamidine resistance gene of Saccharomyces cerevisiae
Journal article   Open access   Peer reviewed

Characterization of the PNT1 pentamidine resistance gene of Saccharomyces cerevisiae

G Ludewig and C Staben
Antimicrobial agents and chemotherapy, Vol.38(12), pp.2850-2856
12/1994
DOI: 10.1128/AAC.38.12.2850
PMCID: PMC188296
PMID: 7695273
url
https://doi.org/10.1128/AAC.38.12.2850View
Published (Version of record) Open Access

Abstract

The Saccharomyces cerevisiae PNT1 gene was isolated and characterized. When present in high copy number in S. cerevisiae, PNT1 confers resistance to the anti-Pneumocystis carinii drug pentamidine. The PNT1 gene encodes a previously uncharacterized polypeptide of 409 amino acids. The predicted gene product is a very basic (pI 9.9) polypeptide with one potential membrane-associated region. PNT1 is located on chromosome XVR of S. cerevisiae. It is transcribed at a very low level. Overexpression of the gene increases resistance to the cytostatic and mitochondrial DNA-damaging effects of pentamidine and related cationic compounds. Disruption of the gene leads to slightly increased levels of susceptibility to pentamidine and some related compounds.
Amino Acid Sequence Drug Resistance - genetics Saccharomyces cerevisiae - genetics Base Sequence Molecular Sequence Data Genes, Fungal Saccharomyces cerevisiae - drug effects Chromosome Mapping Antimycin A - pharmacology Pentamidine - pharmacology

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