Logo image
Osmolyte effects on helix formation in peptides and the stability of coiled-coils
Journal article   Open access   Peer reviewed

Osmolyte effects on helix formation in peptides and the stability of coiled-coils

Scott A Celinski and J Martin Scholtz
Protein science, Vol.11(8), pp.2048-2051
08/2002
DOI: 10.1110/ps.0211702
PMCID: PMC2373673
PMID: 12142459
url
https://europepmc.org/articles/pmc2373673View
Published (Version of record) Open Access

Abstract

The ability of several naturally occurring substances known as osmolytes to induce helix formation in an alanine-based peptide have been investigated. As predicted by the osmophobic effect hypothesis, the osmolytes studies here do induce helix formation. Trimethylamine-N-oxide (TMAO) is the best structure-inducing osmolytes investigated here, but it is not as effective in promoting helix formation as the common cosolvent trifluoroethanol (TFE). We also provide a semiquantitative study of the ability of TMAO to induce helix formation and urea, which acts as a helix (and protein) denaturant. We find that on a molar basis, these agents are exactly counteractive as structure inducing and unfolding agents. Finally, we extend the investigations to the effects of urea and TMAO on the stability of a dimeric coiled-coil peptide and find identical results. Together these results support the tenets of the osmophobic hypothesis and highlight the importance of the polypeptide backbone in protein folding and stability.
Alanine - chemistry Amino Acid Sequence Circular Dichroism Dimerization DNA-Binding Proteins Leucine Zippers - drug effects Methylamines - pharmacology Molecular Sequence Data Osmolar Concentration Protein Denaturation Protein Folding Protein Kinases - chemistry Protein Structure, Secondary - drug effects Saccharomyces cerevisiae Proteins - chemistry Trifluoroethanol - pharmacology Urea - pharmacology

Details

Logo image