Logo image
Thymidine phosphorylase expression in metastatic sites is predictive for response in patients with colorectal cancer treated with continuous oral capecitabine and biweekly oxaliplatin
Journal article   Peer reviewed

Thymidine phosphorylase expression in metastatic sites is predictive for response in patients with colorectal cancer treated with continuous oral capecitabine and biweekly oxaliplatin

Roberto Petrioli, Gianluca Bargagli, Stefano Lazzi, Alessandra Pascucci, Edoardo Francini, Cristiana Bellan, Raffaele Conca, Ignazio Martellucci, Anna Ida Fiaschi, Bruno Lorenzi, …
Anti-cancer drugs, Vol.21(3), pp.313-319
03/2010
DOI: 10.1097/CAD.0b013e328334d88a
PMID: 20016369

View Online

Abstract

The primary objective of this study was to determine the activity and safety profile of biweekly oxaliplatin combined with continuous oral capecitabine in the first-line treatment of metastatic colorectal cancer. A secondary endpoint was to investigate the correlation between thymidylate synthase and thymidine phosphorylase (TP) expression in metastatic tissues and tumor response. Forty-one patients received oral capecitabine 1331 mg/m(2) every day combined with intravenous oxaliplatin 85 mg/m(2) every 2 weeks. The overall response rate was 58.5% [95% confidence interval (CI): 43.3-73.6%], the median progression-free survival 9.4 months ( 95% CI: 7.7-11.2 months) and the median survival 22.3 months (95% CI: 16.1-27.5 months). There were no grade 4 toxicities, and grade 3 toxicity was also uncommon. High TP expression in metastatic tissue was significantly associated with response to treatment (P = 0.019), and also with a trend towards a better median progression-free survival and overall survival compared with patients expressing low TP (P = 0.056; P = 0.073). This study suggests that biweekly oxaliplatin and continuous oral capecitabine is an active and well-tolerated chemotherapy regimen in the first-line treatment of metastatic colorectal cancer. Moreover, these findings add to a growing body of evidence that patients with high levels of intratumoral TP expression are the ideal candidates for capecitabine-based chemotherapy. Anti-Cancer Drugs 21: 313-319 (C) 2010 Wolters Kluwer Health vertical bar Lippincott Williams & Wilkins.
Life Sciences & Biomedicine Oncology Pharmacology & Pharmacy Science & Technology

Details

Metrics

Logo image