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Total Synthesis of the Highly Potent Anti-HIV Natural Product Daurichromenic Acid along with Its Two Chromane Derivatives, Rhododaurichromanic Acids A and B
Journal article   Peer reviewed

Total Synthesis of the Highly Potent Anti-HIV Natural Product Daurichromenic Acid along with Its Two Chromane Derivatives, Rhododaurichromanic Acids A and B

Ying Kang, Yan Mei, Yuguo Du and Zhendong Jin
Organic letters, Vol.5(23), pp.4481-4484
11/01/2003
DOI: 10.1021/ol030109m
PMID: 14602030

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Abstract

(Equation presented) The highly potent anti-HIV natural product daurichromenic acid was successfully synthesized in only five steps with 49% overall yield. The key step in the synthetic strategy involves a microwave-assisted tandem condensation and intramolecular SN2′- type cyclization to form the 2H-benzopyran core structure.

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